December, 2024 | GABAReceptorInhibitorgabareceptorinhibitor

SJ000291942

rofalproject December 21, 2024 0 Comments

Product Name : SJ000291942Description:SJ000291942 is a bone morphogenic protein (BMP) signaling activator.CAS: 425613-09-8Molecular Weight:318.30Formula: C16H15FN2O4Chemical Name: 2-(4-ethylphenoxy)-N-(4-fluoro-3-nitrophenyl)-acetamideSmiles : CCC1C=CC(=CC=1)OCC(=O)NC1=CC(=C(F)C=C1)()=OInChiKey: YSZJLXPXVFGTNK-UHFFFAOYSA-NInChi : InChI=1S/C16H15FN2O4/c1-2-11-3-6-13(7-4-11)23-10-16(20)18-12-5-8-14(17)15(9-12)19(21)22/h3-9H,2,10H2,1H3,(H,18,20)Purity: ≥98% (or refer to the Certificate of Analysis)Shipping…

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LDN-212320

rofalproject December 20, 2024 0 Comments

Product Name : LDN-212320Description:LDN-0212320 Maleate is a novel activator of glutamate transporter EAAT2 translation.CAS: 894002-50-7Molecular Weight:409.46Formula: C21H19N3O4SChemical Name: 3-thio]-6-(2-pyridinyl)-pyridazine maleateSmiles : CC1=CC=CC=C1CSC1=CC=C(N=N1)C1=CC=CC=N1.OC(=O)/C=C\C(O)=OInChiKey: QIGJQEQXFAVIPF-BTJKTKAUSA-NInChi : InChI=1S/C17H15N3S.C4H4O4/c1-13-6-2-3-7-14(13)12-21-17-10-9-16(19-20-17)15-8-4-5-11-18-15;5-3(6)1-2-4(7)8/h2-11H,12H2,1H3;1-2H,(H,5,6)(H,7,8)/b;2-1-Purity: ≥98% (or refer to the…

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NS-6180

rofalproject December 19, 2024 0 Comments

Product Name : NS-6180Description:NS6-180 is a potent KCa3.1 channel blocker (IC50 values are 9, 14 and 15 nM for rat, human and mouse erythrocyte KCa3.1 channels respectively). NS6180 prevents T-cell…

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BI-2536 — PLK1 and BRD4 Dual Inhibitor

rofalproject December 18, 2024 0 Comments

Product Name : BI-2536 --- PLK1 and BRD4 Dual InhibitorDescription:BI-2536 is a potent inhibitor of PLK1 (Polo-like kinase 1, IC50 ~0.83 nM) and BRD4 (IC50 ~37 nM). It also inhibits…

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NLRP3-IN-9

rofalproject December 17, 2024 0 Comments

Product Name : NLRP3-IN-9Description:NLRP3-IN-9 is an inhibitor of caspase-1 and NLRP3 ATPase activities. It acts by irreversibly trapping thiol nucleophiles, which prevents both ATP- and nigericin-triggered pyroptosis of human THP-1…

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10-Hydroxydecanoic acid

rofalproject December 16, 2024 0 Comments

Product Name : 10-Hydroxydecanoic acidDescription:10-Hydroxydecanoic acid (NSC 15139) is a saturated fatty acid of 10-hydroxy-trans-2-decenoic acid from royal jelly, with anti-inflammatory activity.CAS: 1679-53-4Molecular Weight:188.26Formula: C10H20O3Chemical Name: 10-hydroxydecanoic acidSmiles : OCCCCCCCCCC(O)=OInChiKey:…

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1-Pentadecanol

rofalproject December 15, 2024 0 Comments

Product Name : 1-PentadecanolDescription:1-Pentadecanol is a naturally occurring antiacne agent.CAS: 629-76-5Molecular Weight:228.41Formula: C15H32OChemical Name: pentadecan-1-olSmiles : CCCCCCCCCCCCCCCOInChiKey: REIUXOLGHVXAEO-UHFFFAOYSA-NInChi : InChI=1S/C15H32O/c1-2-3-4-5-6-7-8-9-10-11-12-13-14-15-16/h16H,2-15H2,1H3Purity: ≥98% (or refer to the Certificate of Analysis)Shipping Condition: Shipped…

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2OH-BNPP1

rofalproject December 14, 2024 0 Comments

Product Name : 2OH-BNPP1Description:2OH-BNPP1 is an inhibitor of BUB1 kinase, a Ser/Thr kinase, used for the treatment of cancer.CAS: 833481-73-5Molecular Weight:297.35Formula: C16H19N5OChemical Name: 2-({4-amino-1-tert-butyl-1H-pyrazolopyrimidin-3-yl}methyl)phenolSmiles : CC(C)(C)N1N=C(CC2=CC=CC=C2O)C2=C(N)N=CN=C12InChiKey: LWLCFWPPMNPMOI-UHFFFAOYSA-NInChi : InChI=1S/C16H19N5O/c1-16(2,3)21-15-13(14(17)18-9-19-15)11(20-21)8-10-6-4-5-7-12(10)22/h4-7,9,22H,8H2,1-3H3,(H2,17,18,19)Purity: ≥98%…

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Dasatinib metabolite M6

rofalproject December 13, 2024 0 Comments

Product Name : Dasatinib metabolite M6Description:Dasatinib metabolite M6 (Dasatinib carboxylic acid) is an oxidative metabolite of Dasatinib (HY-10181). Dasatinib is a potent and orally active dual Bcr-Abl and Src family…

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CMP-5 hydrochloride

rofalproject December 13, 2024 0 Comments

Product Name : CMP-5 hydrochlorideDescription:CMP-5 hydrochloride is a potent, specific, and selective PRMT5 inhibitor, while displays no activity against PRMT1, PRMT4, and PRMT7 enzymes. CMP-5 hydrochloride selectively blocks S2Me-H4R3 by…

SJ000291942

LDN-212320

NS-6180

BI-2536 — PLK1 and BRD4 Dual Inhibitor

NLRP3-IN-9

10-Hydroxydecanoic acid

1-Pentadecanol

2OH-BNPP1

Dasatinib metabolite M6

CMP-5 hydrochloride

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