6-Iodonordihydrocapsaicin
Product Name : 6-IodonordihydrocapsaicinDescription:IC50: 10 nm against 100 nm capsaicin The vanilloid TRPV1 receptor, also known as VR1 receptor, belongs to the large family of ‘transient receptor potential’ (TRP). TRPV1…
Methiothepin maleate
Product Name : Methiothepin maleateDescription:Methiothepin is a non-selective antagonist of the serotonin (5-HT) receptor. It is a potent antagonist of 5-HT1A and 5-HT1B (IC50 = 16 nM and Ki =…
Eticlopride hydrochloride
Product Name : Eticlopride hydrochlorideDescription:Product informationCAS: 97612-24-3Molecular Weight:377.31Formula: C17H26Cl2N2O3Chemical Name: (1R,2S)-2-{methyl}-1-ethylpyrrolidin-1-ium chlorideSmiles : .COC1C(Cl)=CC(CC)=C(O)C=1C(=O)NC1CCC1CCInChiKey: HFJFXXDHVWLIKX-YDALLXLXSA-NInChi : InChI=1S/C17H25ClN2O3.ClH/c1-4-11-9-13(18)16(23-3)14(15(11)21)17(22)19-10-12-7-6-8-20(12)5-2;/h9,12,21H,4-8,10H2,1-3H3,(H,19,22);1H/t12-;/m0./s1Purity: ≥98% (or refer to the Certificate of Analysis)Shipping Condition: Shipped under ambient temperature…
Acifran
Product Name : AcifranDescription:Product informationCAS: 72420-38-3Molecular Weight:218.21Formula: C12H10O4Chemical Name: (5R)-5-methyl-4-oxo-5-phenyl-4,5-dihydrofuran-2-carboxylic acidSmiles : C1(OC(=CC1=O)C(O)=O)C1C=CC=CC=1InChiKey: DFDGRKNOFOJBAJ-GFCCVEGCSA-NInChi : InChI=1S/C12H10O4/c1-12(8-5-3-2-4-6-8)10(13)7-9(16-12)11(14)15/h2-7H,1H3,(H,14,15)/t12-/m1/s1Purity: ≥98% (or refer to the Certificate of Analysis)Shipping Condition: Shipped under ambient temperature as…
[Orn5]-URP
Product Name : -URPDescription:-URP is a potent and selective pure antagonist of Urotensin-II receptor (UT), with an pEC50 of 7.24. -URP displays no agonist activity.CAS: 782485-03-4Molecular Weight:1003.20Formula: C48H62N10O10S2Chemical Name: (2S)-2-amino]-10-(3-aminopropyl)-16-benzyl-6,9,12,15,18-pentahydroxy-7--13--1,2-dithia-5,8,11,14,17-pentaazacycloicosa-5,8,11,14,17-pentaen-4-yl](hydroxy)methylidene}amino]-3-methylbutanoic…
Eurycomalactone
Product Name : EurycomalactoneDescription:Eurycomalactone is a natural product found in Eurycoma longifolia Jack., acts as a potent NF-κB inhibitor, with an IC50 of 0.5 μM. Eurycomalactone inhibits protein synthesis, depletes…
Licoflavone B
Product Name : Licoflavone BDescription:Licoflavone B is a flavonoid isolated from Glycyrrhiza inflata, inhibits S. mansoni ATPase (IC50, 23.78 µM) and ADPase (IC50, 31.50 µM) activity. Anti-schistosomiasis activity.CAS: 91433-17-9Molecular Weight:390.47Formula:…
Medicagenic acid
Product Name : Medicagenic acidDescription:Medicagenic acid (Castanogenin) is isolated from the roots of Herniaria glabra L, exhibits potent fungistatic effects against several plant pathogens and human dermatophytes. Medicagenic acid (Castanogenin)…
GSK2850163
Product Name : GSK2850163Description:GSK2850163 is a novel inhibitor of inositol-requiring enzyme-1 alpha (IRE1α) which can inhibit IRE1α kinase activity and RNase activity with IC50s of 20 and 200 nM, respectively.CAS:…
FAAH-IN-1
Product Name : FAAH-IN-1Description:FAAH-IN-1 is a fatty acid amide hydrolase (FAAH) inhibitor, with IC50s of 145 nM and 650 nM for rat and human FAAH, respectively.CAS: 1242441-47-9Molecular Weight:398.91Formula: C20H19ClN4OSChemical Name:…